Synthesis of Heterocyclic Dipeptide Analogues.
نویسندگان
چکیده
منابع مشابه
Synthesis and modifications of phosphinic dipeptide analogues.
Pseudopeptides containing the phosphinate moiety (-P(O)(OH)CH(2)-) have been studied extensively, mainly as transition state analogue inhibitors of metalloproteases. The key synthetic aspect of their chemistry is construction of phosphinic dipeptide derivatives bearing appropriate side-chain substituents. Typically, this synthesis involves a multistep preparation of two individual building bloc...
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Benzo-condensed four-ring heterocycles, such as benzoxetes 1 and benzothietes 3 represent multi-purpose starting compounds for the preparation of various higher heterocyclic ring systems. The thermal or photochemical valence isomerizations between the benzenoid forms 1,3 and the higher reactive o-quinoid structures 2,4 provide the basis for the synthetic applications. On the other hand, this va...
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ژورنال
عنوان ژورنال: Acta Chemica Scandinavica
سال: 1998
ISSN: 0904-213X
DOI: 10.3891/acta.chem.scand.52-1327